发明名称 SYNTHESIS OF CHIRALLY PURIFIED SUBSTITUTED BENZOTHIAZOLE DIAMINES
摘要 Methods for preparing chirally purified substituted 4,5,6,7-tetrahydro-benzotiazole diamines such as, for example, (6R)2-amino-4,5,6,7-tetrahydro-6-(propylamino)benzothiazole and purifying a dominant enantiomer of substituted 4,5,6,7-tetrahydro-benzotiazole diamines from entantiomerically enriched mixtures of substituted 4,5,6,7-tetrahydro-benzotiazole diamines are provided herein.
申请公布号 WO2008113056(A2) 申请公布日期 2008.09.18
申请号 WO2008US57158 申请日期 2008.03.14
申请人 KNOPP NEUROSCIENCES, INC.;RAJE, PRASAD;GADIKOTA, RAJENDRAKUMAR, REDDY;CHEN, JIAN-XIE;LAPINA, OLGA;MCCALL, JOHN, M. 发明人 RAJE, PRASAD;GADIKOTA, RAJENDRAKUMAR, REDDY;CHEN, JIAN-XIE;LAPINA, OLGA;MCCALL, JOHN, M.
分类号 C07D277/82 主分类号 C07D277/82
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