发明名称 |
SYNTHESIS OF CHIRALLY PURIFIED SUBSTITUTED BENZOTHIAZOLE DIAMINES |
摘要 |
Methods for preparing chirally purified substituted 4,5,6,7-tetrahydro-benzotiazole diamines such as, for example, (6R)2-amino-4,5,6,7-tetrahydro-6-(propylamino)benzothiazole and purifying a dominant enantiomer of substituted 4,5,6,7-tetrahydro-benzotiazole diamines from entantiomerically enriched mixtures of substituted 4,5,6,7-tetrahydro-benzotiazole diamines are provided herein. |
申请公布号 |
WO2008113056(A2) |
申请公布日期 |
2008.09.18 |
申请号 |
WO2008US57158 |
申请日期 |
2008.03.14 |
申请人 |
KNOPP NEUROSCIENCES, INC.;RAJE, PRASAD;GADIKOTA, RAJENDRAKUMAR, REDDY;CHEN, JIAN-XIE;LAPINA, OLGA;MCCALL, JOHN, M. |
发明人 |
RAJE, PRASAD;GADIKOTA, RAJENDRAKUMAR, REDDY;CHEN, JIAN-XIE;LAPINA, OLGA;MCCALL, JOHN, M. |
分类号 |
C07D277/82 |
主分类号 |
C07D277/82 |
代理机构 |
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代理人 |
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地址 |
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