发明名称 |
Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |
摘要 |
Disclosed are cyclopentyl compounds linked to a benzoxazinyl group through an amido moiety utilising the ring nitrogen of the benzoxazine. In particular disclosed are compounds of formula I wherein the substituents are described in the specification, useful as modulators of chemokine receptors. These compounds can be used in the treatment, amelioration, control or reduction of risk of an inflammatory and immunoregulatory disorders or diseases.
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申请公布号 |
NZ543287(A) |
申请公布日期 |
2008.08.29 |
申请号 |
NZ20040543287 |
申请日期 |
2004.04.08 |
申请人 |
MERCK & CO., INC. |
发明人 |
GOBLE, STEPHEN D;MILLS, SANDER G;YANG, LIHU;PASTERNAK, ALEXANDER |
分类号 |
A61K;A61K31/535;A61K31/55;A61P29/00;C07D;C07D243/00;C07D265/12;C07D401/00;C07D413/00;C07D413/08;C07D413/14;C07D417/00;C07D417/14;C07D498/04;C07D519/00;(IPC1-7):A61P29/00 |
主分类号 |
A61K |
代理机构 |
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主权项 |
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地址 |
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