发明名称 HETEROCYCLIC DERIVATIVES AS M3 MUSCARINIC RECEPTORS
摘要 This invention relates to M3 antagonists of formula (I) wherein R<SUP>2</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, R<SUP>6</SUP>, W, V, A, D, X, t, u and v are as defined herein; pharmaceutical compositions containing them; methods for their preparation; and their use in the treatment of diseases where enhanced M3 receptor activation is implicated.
申请公布号 WO2008099186(A1) 申请公布日期 2008.08.21
申请号 WO2008GB00519 申请日期 2008.02.14
申请人 ARGENTA DISCOVERY LIMITED;AVITABILE, BARBARA, GIUSEPPINA;FINCH, HARRY;KNIGHT, JAMIE, DAVID;NADIN, ALAN, JOHN;RAY, NICHOLAS, CHARLES 发明人 AVITABILE, BARBARA, GIUSEPPINA;FINCH, HARRY;KNIGHT, JAMIE, DAVID;NADIN, ALAN, JOHN;RAY, NICHOLAS, CHARLES
分类号 C07D471/08;A61K31/439;A61P1/00;A61P9/00;A61P11/00 主分类号 C07D471/08
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