发明名称 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS
摘要 This invention is directed to pyridopyrimidinone compounds of formula (I): wherein n, R<SUP>1</SUP>, R<SUP>2 </SUP>and R<SUP>3 </SUP>are as defined herein, as a stereoisomer, enantiomer, tautomer thereof or mixtures thereof; or a pharmaceutically acceptable salt, solvate or prodrug thereof, useful for the treatment and/or prevention of sodium channel-mediated diseases or conditions, such as pain.
申请公布号 US2008194616(A1) 申请公布日期 2008.08.14
申请号 US20080026435 申请日期 2008.02.05
申请人 XENON PHARMACEUTICALS INC. 发明人 LIU SHIFENG;FU JIANMIN;KAMBOJ RAJENDER;CHOWDHURY SULTAN;JIA QI;WOOD MARK;SUN JIANYU
分类号 A61K31/444;A61P29/00;C07D471/02 主分类号 A61K31/444
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