发明名称 IBANDRONATE SODIUM PROPYLENE GLYCOL SOLVATE AND PROCESSES FOR THE PREPARATION THEREOF
摘要 <p>Ibandronate sodium and propylene glycol readily forms a free-flowing crystalline solvate. The novel solvate is non-hygroscopic, free-flowing, chemically and polymorphically stable, and easily dried even on industrial scale. Thus, it is particularly suitable for pharmaceutical applications. A process for preparing said novel solvate is further disclosed. Formula (I).</p>
申请公布号 WO2008070960(A1) 申请公布日期 2008.06.19
申请号 WO2007CA02093 申请日期 2007.11.21
申请人 APOTEX PHARMACHEM INC.;REY, ALLAN, W.;STRADIOTTO, DAVID, A.;DATTA, PROBAL, KANTI;TRAYNOR, KRISTA, LYN;MCPHAIL, CAMERON, L. 发明人 REY, ALLAN, W.;STRADIOTTO, DAVID, A.;DATTA, PROBAL, KANTI;TRAYNOR, KRISTA, LYN;MCPHAIL, CAMERON, L.
分类号 C07F9/38;A61K31/663;A61P19/10 主分类号 C07F9/38
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