发明名称 RETROVIRAL PROTEASE INHIBITING COMPOUND
摘要 PROBLEM TO BE SOLVED: To provide a new compound as an HIV protease inhibiting compound, and to provide a production intermediate thereof. SOLUTION: A compound represented by formula (1) is provided. Wherein, R1 and R2 are independently selected from the group consisting of an alkyl, a cycloalkyl and an arylalkyl; R3 is a lower alkyl, a hydroxyalkyl, or a cycloalkylalkyl; R4 is an aryl or a heterocycle; R5 is a 5-7 membered ring containing nitrogen atom and having a hetero atom directly bonded with the heterocycle; and L1 is a bivalent bonding group such as -O- or -S-. COPYRIGHT: (C)2008,JPO&INPIT
申请公布号 JP2008115189(A) 申请公布日期 2008.05.22
申请号 JP20070327351 申请日期 2007.12.19
申请人 ABBOTT LAB 发明人 SHAM HING LEUNG;NORBECK DANIEL W;CHEN XIAOQI;BETEBENNER DAVID A;DALE J KEMP;THOMAS R HERIN;GONDEI N KUMAA;STEVEN L CONDON;ARTHUR J COOPER;DANIEL A DICKMAN;STEVEN M HANNIKKU;LAWRENCE KORATSUEKOUSUKII;PATRICIA A OLIVER;DANIEL J PRATA;PETER J STENGEL;ERIK J SUTOONAA;JII-HAA J TEIEN;JII-HOWA RIU;KETAN M PATEL
分类号 C07D207/27;C07D253/00;A61K31/00;A61K31/40;A61K31/4015;A61K31/41;A61K31/415;A61K31/4164;A61K31/4166;A61K31/4178;A61K31/4184;A61K31/42;A61K31/421;A61K31/425;A61K31/427;A61K31/4427;A61K31/443;A61K31/4433;A61K31/4439;A61K31/47;A61K31/495;A61K31/496;A61K31/4965;A61K31/505;A61K31/506;A61K31/513;A61K31/53;A61K31/55;A61K38/05;A61K45/00;A61P31/18;A61P43/00;C07C231/12;C07C235/20;C07C273/18;C07C275/16;C07D;C07D207/22;C07D207/26;C07D207/273;C07D207/34;C07D207/40;C07D207/404;C07D207/408;C07D207/416;C07D211/72;C07D211/84;C07D223/06;C07D233/28;C07D233/30;C07D233/32;C07D233/34;C07D233/36;C07D233/40;C07D233/42;C07D233/66;C07D239/06;C07D239/10;C07D239/20;C07D239/22;C07D241/06;C07D241/08;C07D241/18;C07D243/04;C07D253/06;C07D263/16;C07D263/20;C07D263/22;C07D263/34;C07D265/04;C07D267/04;C07D277/12;C07D277/32;C07D277/34;C07D279/06;C07D281/02;C07D401/12;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12 主分类号 C07D207/27
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