发明名称 METHOD FOR PRODUCING 4(3H)-QUINAZOLINONE DERIVATIVE
摘要 <p>This invention is related to a method for producing 3-{4-[3-(1-pyrrolidinyl)propoxy]phenyl}-5-trifluoromethyl-4(3H)-quinazolinone comprising a step for reacting 2-methyl-5-trifluoromethyl-4H-3,1-benzoxazin-4-one with 4-[3-(1-pyrrolidinyl)propoxy]aniline or an acid-addition salt thereof, or 4-(1-cyclobutyl-4-piperidiny9oxyaniline or acid addition salt thereof in the presence of an acid catalyst.</p>
申请公布号 EP1903040(A1) 申请公布日期 2008.03.26
申请号 EP20060780913 申请日期 2006.07.04
申请人 BANYU PHARMACEUTICAL CO., LTD.;MERCK & CO., INC. 发明人 SAWADA, NAOTAKA;TSURITANI, TAKAYUKI;SATO, KIMIHIKO;ITOH, TAKAHIRO;AKAO, ATSUSHI;KADOWAKI, CHIE;IIDA, TAKEHIKO;YASUDA, NOBUYOSHI;MASE, TOSHIAKI
分类号 C07D403/12 主分类号 C07D403/12
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