发明名称 STABLE C-GLYCOSIDE SUGAR AND C-GLYCOCONJUGATE MIMETICS, METHOD FOR PREPARING SAME AND USES THEREOF IN PARTICULAR IN COSMETICS AND DRUGS
摘要 The invention concerns a C-glycoside compound of formula (I); wherein: n is equal to 1 or 2; Y represents H or halogen; X is an alkyl chain bearing at least one amino, amide, acid, ester, carbonyl, alcohol, aryl function or a carbonyl, ester amide, amino, alcohol group; the R's, identical or different, represent a OH or OR' group where R' is an alkyl, benzyl, benzoyl, acetyl, pivaloyl, trialkylsilyl, tertiobutyldiphenylsilyl group or one or more sugars; R1 represents OR', NR"R'", N3, or a phthalamide with R'' and R''', identical or different, represent H or an alkyl, aryl, benzyl, benzoyl, acetyl, alkoxycarbonyl, allyloxycarbonyl, benzyloxycarbonyl group; R2 represents H or halogen or a OH, OR, NR"R"'or N3 group, as well as derivatives thereof in physiologically or pharmaceutically acceptable base, mineral or organic acid-addition salt, hydrate or solvate form. The invention is useful for preparing C-glycoside compounds or C-glycoconjugates applicable in particular in cosmetology, medical imagery, immunology for treating cancer, diabetes, hypertension.
申请公布号 WO2007128899(A3) 申请公布日期 2008.03.13
申请号 WO2007FR00683 申请日期 2007.04.23
申请人 INSTITUT NATIONAL DES SCIENCES APPLIQUEES DE ROUEN (INSA);CASTELOT-DELIENCOURT-GODEFROY, GERALDINE;QUIRION, JEAN-CHARLES;JUBAULT, PHILIPPE;ZOUTE, LUDIVINE 发明人 CASTELOT-DELIENCOURT-GODEFROY, GERALDINE;QUIRION, JEAN-CHARLES;JUBAULT, PHILIPPE;ZOUTE, LUDIVINE
分类号 C07H7/00;C07D307/20;C07D307/32;C07D309/10;C07D309/30 主分类号 C07H7/00
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