发明名称 BETA-CARBOLINES USEFUL FOR TREATING INFLAMMATORY DISEASE
摘要 This invention provides beta-carboline compounds of formula (I) wherein Ring A is a substituted pyridinyl, pyrimidinyl, morpholinyl, piperidinyl, piperazinyl, pyrrolidinyl, pyranyl, tetrahydrofuranyl, cyclohexyl, cyclopentyl or thiomorpholinyl ring and R1, R2 and R3 are as described in the specification. The compounds are IKK-2 inhibitors that are useful for treating IKK-2 mediated diseases such as inflammatory diseases and cancer.
申请公布号 RS20050832(A) 申请公布日期 2007.12.31
申请号 YUP20050832 申请日期 2004.04.09
申请人 MILLENNIUM PHARMACEUTICALS,INC. 发明人 HEPPERLE MICHAEL;LIU JULIE FIELDS;SOUCY FRANCOIS;YE YINGCHUN;MURRAY ROBERT;PRAKASH RAMAN;LITTLE JEREMY;CASTRO ALFREDO;MAZDIYASNI HORMOZ;FLEMING PAUL;REYNOLDS DOMINIC
分类号 C07D471/04;A61K31/437;C07D265/30 主分类号 C07D471/04
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