发明名称 2-Iminopyrrolidine derivatives
摘要 A 2-iminoimidazole derivative represented by the formula: <CHEM> äwherein R<1>, R<2> and R<3> represent hydrogen, optionally substituted C1-6 alkyl, etc.; R<6> represents hydrogen, C1-6 alkyl, C1-6 alkyloxycarbonyl, etc.; Y<1> represents a single bond, -CH2-, etc.; Y<2> represents a single bond, -CO-, etc.; and Ar represents hydrogen, a group represented by the formula: <CHEM> Äwherein R<10>-R<14> represent hydrogen, C1-6 alkyl, hydroxyl, C1-6 alkoxy, etc., and R<11> and R<12> or R<12> and R<13> may bond together to form a 5- to 8-membered heterocycleÜ, etc.ü or a salt thereof.
申请公布号 AU2005202135(B2) 申请公布日期 2007.11.15
申请号 AU20050202135 申请日期 2005.05.17
申请人 EISAI R AND D MANAGEMENT CO., LTD. 发明人 SHUICHI SUZUKI;AKIFUMI KIMURA;ATSUSHI KAMADA;MAKOTO KOTAKE;IEHARU HISHINUMA;YOSHIMITSU NAOE;TAKASHI MUSHA;MASANOBU SHINODA;MOTOJI KOGUSHI;KEN-ICHI CHIBA;YOSHIAKI OOHASHI;KAZUO OKANO;HIROSHI TANAKA;HIROKO KOBAYASHI;RICHARD CLARK;TOSHIYUKI MATSUOKA;NAOTO ONO;FUMIHIRO OZAKI;ITARU TSUKADA;SYUHEI MIYAZAWA;NOBUAKI SATO;TSUTOMU KAWATA;TETSUYA KAWAHARA;MITSUAKI MIYAMOTO;TARO TERAUCHI;OSAMU ITO;FUMIYOSHI MATSUURA;AKIHARU KAJIWARA
分类号 C07D209/44;A61K31/403;A61K31/4035;A61K31/4178;A61K31/4184;A61K31/422;A61K31/437;A61K31/454;A61K31/496;A61K31/5377;A61K31/538;A61P7/02;A61P9/00;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/12;A61P19/10;A61P25/00;A61P29/00;A61P35/00;A61P43/00;C07D209/62;C07D401/10;C07D403/06;C07D403/10;C07D405/06;C07D413/06;C07D471/04 主分类号 C07D209/44
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