发明名称 HETEROCYCLIC DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF
摘要 The invention concerns compounds of formula (I) wherein: X represents a -C-, -SO<SUB>2</SUB>-, -C-N(R<SUB>5</SUB>)-C-N(R<SUB>5</SUB>)- group; Y represents an oxygen atom or a sulphur atom; R<SUB>1</SUB> represents a hydrogen atom or a C<SUB>1</SUB>-C<SUB>4</SUB> alkyl group; R<SUB>2</SUB> represents a C<SUB>1</SUB>-C<SUB>7</SUB> alkyl group, a carbocyclic radical, a methyl substituted by a C<SUB>3</SUB>-C<SUB>12</SUB> non aromatic carbocyclic radical, a phenyl, a phenoxymethyl, a benzyl, a benzhydryl, a benzhydrylmethyl group, a 1,2,3,4-tetrahydronaphthalenyl, a pyrrolyl, imidazolyl, pyridyl, pyrazolyl, furyl, thienyl radical; an indolyl; a benzofuryl; R<SUB>3</SUB> represents a substituted or unsubstituted phenyl; R<SUB>4</SUB> represents a substituted or unsubstituted phenyl; R<SUB>5</SUB> represents a hydrogen atom or a C<SUB>1</SUB>-C<SUB>4</SUB> alkyl; as well as their salts and solvates. The invention also concerns a method for preparing same and the therapeutic use thereof.
申请公布号 WO2007068815(A3) 申请公布日期 2007.11.01
申请号 WO2006FR02695 申请日期 2006.12.11
申请人 SANOFI-AVENTIS;BARTH, FRANCIS;RINALDI-CARMONA, MURIELLE 发明人 BARTH, FRANCIS;RINALDI-CARMONA, MURIELLE
分类号 C07D277/28;A61K31/421;A61K31/426;A61K31/427;A61P25/32;A61P29/00;C07D263/32;C07D417/12 主分类号 C07D277/28
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