发明名称 METHOD FOR PRODUCING 4-ALKOXYPYRIDINE-1-OXIDE DERIVATIVE
摘要 PROBLEM TO BE SOLVED: To provide a method for producing a 4-alkoxypyridine-1-oxide derivative used as an intermediate for producing benzimidazole derivatives useful as gastric inhibitory agents and antiulcer agents in excellent workability and in excellent operability in a state free from the risk of explosion. SOLUTION: This method for producing the 4-alkoxypyridine-1-oxide derivative represented by formula (I) (Ra and Rc are each H or the like; W is a single bond or the like; Rb is a 1 to 6C alkyl or the like) is characterized by comprising a process for reacting a pyridine-N-oxide derivative with a compound of HO-W-Rb in the presence of potassium hydroxide in toluene. COPYRIGHT: (C)2008,JPO&INPIT
申请公布号 JP2007284372(A) 申请公布日期 2007.11.01
申请号 JP20060112340 申请日期 2006.04.14
申请人 EISAI R & D MANAGEMENT CO LTD 发明人 SUGANO GORO
分类号 C07D405/12 主分类号 C07D405/12
代理机构 代理人
主权项
地址