| 发明名称 |
Process for the preparation of perindopril |
| 摘要 |
A process for preparing perindopril (III) or a pharmaceutically acceptable salt thereof, which process comprises a substituted benzyl ester of (2S,3aS,7aS)-octahydroindole-2-carboxylic acid (I) with N-[(S)-carbethoxybutyl]-(S)-alanine (II) where R represents a halo, C<SUB>1-4 </SUB>alkoxy or nitro substituent. |
| 申请公布号 |
US2007185335(A1) |
申请公布日期 |
2007.08.09 |
| 申请号 |
US20050599918 |
申请日期 |
2005.04.07 |
| 申请人 |
KANKAN RAJENDRA N;RAO DHARMARAJ R |
发明人 |
KANKAN RAJENDRA N.;RAO DHARMARAJ R. |
| 分类号 |
C07D209/02;C07D209/42;C07K5/06 |
主分类号 |
C07D209/02 |
| 代理机构 |
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代理人 |
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| 主权项 |
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| 地址 |
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