发明名称 THIAZOLE COMPOUNDS AND METHODS OF USE
摘要 The invention relates to thiazole compounds of Formula (I) and Formula (II) and compositions thereof useful for treating diseases mediated by protein kinase B (PKB) where the variables have the definitions provided herein. The invention also relates to the therapeutic use of such thiazole compounds and compositions thereof in treating disease states associated with abnormal cell growth, cancer, inflammation, and metabolic disorders.
申请公布号 WO2007084391(A2) 申请公布日期 2007.07.26
申请号 WO2007US00871 申请日期 2007.01.11
申请人 AMGEN INC.;ZENG, QINGPING;ALLEN, JOHN G.;BOURBEAU, MATTHEW P.;DOMINGUEZ, CELIA;FOTSCH, CHRISTOPHER H.;HAN, NIANHE;HONG, FANG-TSAO;HUANG, XIN;LEE, MATTHEW R.;LI, AIWEN;LIU, QINGYIAN;RIDER, JAMES T.;TADESSE, SEIFU;TASKER, ANDREW S.;VISWANADHAN, VELLARKAD N.;WANG, XIANGHONG;WEILER, KURT E.;WOHLHIETER, GEORGE E.;YAO, GUOMIN;YUAN, CHESTER CHENGUANG 发明人 ZENG, QINGPING;ALLEN, JOHN G.;BOURBEAU, MATTHEW P.;DOMINGUEZ, CELIA;FOTSCH, CHRISTOPHER H.;HAN, NIANHE;HONG, FANG-TSAO;HUANG, XIN;LEE, MATTHEW R.;LI, AIWEN;LIU, QINGYIAN;RIDER, JAMES T.;TADESSE, SEIFU;TASKER, ANDREW S.;VISWANADHAN, VELLARKAD N.;WANG, XIANGHONG;WEILER, KURT E.;WOHLHIETER, GEORGE E.;YAO, GUOMIN;YUAN, CHESTER CHENGUANG
分类号 C07D417/04;C07D277/42;C07D277/54;C07D417/14;C07D471/04;C07D495/04;C07D513/04 主分类号 C07D417/04
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