发明名称 POLYCYCLIC INDAZOLE DERIVATIVES THAT ARE ERK INHIBITORS
摘要 <p>Disclosed are the ERK inhibitors of formula 1.0 and the pharmaceutically acceptable salts and solvates thereof. Q is a piperidine or piperazine ring that can have a bridge or a fused ring. The piperidine ring can have a double bond in the ring. All other substitutents are as defined herein. Also disclosed are methods of treating cancer using the compounds of formula 1.0.</p>
申请公布号 WO2007070398(A1) 申请公布日期 2007.06.21
申请号 WO2006US46959 申请日期 2006.12.11
申请人 SCHERING CORPORATION;COOPER, ALAN;DENG, YONGQI;SHIPPS, GERALD, W., JR.;SHIH, NENG-YANG;ZHU, HUGH;SUN, ROBERT;KELLY, JOSEPH;DOLL, RONALD;NAN, YANG;WANG, TONG;DESAI, JAGDISH;WANG, JAMES;DONG, YOUHAO;MADISON, VINCENT, S.;LI, XIAO;HRUZA, ALAN;SIDDIQUI, M., ARSHAD;SAMATAR, AHMED;PALIWAL, SUNIL;TSUI, HON-CHUNG;CELEBI, AZIM, A.;WU, YIJI;BOGA, SOBHANA, BABU 发明人 COOPER, ALAN;DENG, YONGQI;SHIPPS, GERALD, W., JR.;SHIH, NENG-YANG;ZHU, HUGH;SUN, ROBERT;KELLY, JOSEPH;DOLL, RONALD;NAN, YANG;WANG, TONG;DESAI, JAGDISH;WANG, JAMES;DONG, YOUHAO;MADISON, VINCENT, S.;LI, XIAO;HRUZA, ALAN;SIDDIQUI, M., ARSHAD;SAMATAR, AHMED;PALIWAL, SUNIL;TSUI, HON-CHUNG;CELEBI, AZIM, A.;WU, YIJI;BOGA, SOBHANA, BABU
分类号 C07D231/56;A61K31/427;A61K31/428;A61K31/496;A61K31/506;A61P35/00;C07D403/12;C07D403/14;C07D409/12;C07D413/12;C07D417/12;C07D417/14 主分类号 C07D231/56
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