发明名称 |
4-substituted or unsubstituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid derivatives as beta-lactamase inhibitors |
摘要 |
The present invention relates to novel, low molecular weight broad spectrum compounds in particular to a class of 4-substituted or unsubstituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid or their derivatives which have beta-lactamase inhibitory and antibacterial properties. The compounds are therefore useful in the treatment of antibacterial infections in humans or animals, either alone or in combination with other antibiotics.
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申请公布号 |
US7229983(B2) |
申请公布日期 |
2007.06.12 |
申请号 |
US20040834301 |
申请日期 |
2004.04.28 |
申请人 |
WYETH HOLDINGS CORPORATION |
发明人 |
MANSOUR TAREK SUHAYL;VENKATESAN ARANAPAKAM MUDUMBAI |
分类号 |
A61P31/04;A61K31/55;A61K31/554;C07D281/10;C07D417/02;C07D487/04;C07D498/04 |
主分类号 |
A61P31/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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