发明名称 |
CLASS IIA HISTONE DEACETYLASE (HDAC) SUBSTRATE |
摘要 |
The present invention relates to the use of trifluoroacetylated lysine (Boc-L-Lys(e- trifluoroacetyl)-MCA) as a substrate for histone deacetylases, specific for the class Ha subtype. |
申请公布号 |
WO2007029037(A3) |
申请公布日期 |
2007.05.18 |
申请号 |
WO2006GB50276 |
申请日期 |
2006.09.05 |
申请人 |
ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA;JONES, PHILIP;STEINKUHLER, CHRISTIAN |
发明人 |
JONES, PHILIP;STEINKUHLER, CHRISTIAN |
分类号 |
C12Q1/44;C07D277/56;C07D333/34;C07D333/38;C07D409/08;C07D409/12;C07D409/14;C07D413/12;C07D413/14;C07D417/12;C07D417/14;C07D471/04;C07D471/18;C07D487/04;C07D487/08;C07D487/18;C07D491/10;C07D495/04;C12Q1/34 |
主分类号 |
C12Q1/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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