| 发明名称 |
Ethynyl derivatives serving as factor Xa inhibitors |
| 摘要 |
Novel compounds of the formula (I), in which R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, X and Y have the meaning indicated in Patent claim 1, are inhibitors of coagulation factor Xa and can be employed for the prophylaxis and/or therapy of thromboembolic diseases and for the treatment of tumors. |
| 申请公布号 |
ZA200507818(B) |
申请公布日期 |
2007.02.28 |
| 申请号 |
ZA20050007818 |
申请日期 |
2005.09.27 |
| 申请人 |
MERCK PATENT GMBH. |
发明人 |
MEDERSKI, WERNER;DORSCH, DIETER;GLEITZ, JOHANNES;TSAKLAKIDIS, CHRISTOS;CEZANNE, BERTRAM;VAN AMSTERDAM, CHRISTOPH |
| 分类号 |
A61K;A61P;A61P7/02;C07D;C07D213/64;C07D233/46;C07D265/32;C07D401/12;C07D403/12;C07F;C07F9/6533 |
主分类号 |
A61K |
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