发明名称 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS
摘要 Novel pyrrazole derivative compounds and their use as pharmaceutical agents, in particular their use as TGF-beta signal transduction inhibitors. The disclosed invention relates to compounds of the structure (I) wherein (I) is a four, five, or six membered saturated ring and X is C, O or S.
申请公布号 EA007782(B1) 申请公布日期 2007.02.27
申请号 EA20030001289 申请日期 2002.05.13
申请人 ELI LILLY AND COMPANY 发明人 SAWYER JASON, SCOTT;BEIGHT DOUGLAS, WADE;CIAPETTI PAOLA;DECOLLO TODD, VIVCENT;GODFREY ALEXANDER, GLENN;GOODSON THEODORE, JR.;HERRON DAVID, KENT;LI HONG-YU;LIAO JUNKAI;MCMILLEN WILLIAM, THOMAS;MILLER SHAWN, CHRISTOPHER;MORT NICOLAS, ANTHONY;YINGLING JONATHAN, MICHAEL;SMITH EDWARD, C., R.
分类号 C07D487/04;A61K31/33;A61K31/41;A61K31/4439;A61K31/444;A61K31/4709;A61K31/496;A61K31/535;A61K31/5383;A61K31/55;A61K45/00;A61P3/10;A61P7/04;A61P9/10;A61P13/12;A61P17/02;A61P17/12;A61P19/02;A61P21/02;A61P25/28;A61P27/02;A61P29/00;A61P31/00;A61P31/18;A61P35/00;A61P37/02;A61P37/08;A61P43/00;C07D401/12;C07D471/04;C07D498/04 主分类号 C07D487/04
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