发明名称 |
UREA ANTAGONISTS OF P2Y1. |
摘要 |
<p>The present invention provides novel pyridyl or phenyl ureas and analogues thereof, which are selective inhibitors of the human P2Y1 receptor. The invention also provides for various pharmaceutical compositions of the same and methods for treating diseases responsive to modulation of P2Y1 receptor activity.</p> |
申请公布号 |
MXPA06013022(A) |
申请公布日期 |
2007.01.23 |
申请号 |
MX2006PA13022 |
申请日期 |
2005.05.11 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY. |
发明人 |
REJEAN RUEL.;R. MICHAEL LAWRENCE;HUJI TUERDI;HANNGUANG J. CHAO;JENNIFER X. QIAO;TAMMY C. WANG;TIMUR GUNGOR;TIMOTHY HERPIN;JACQUES YVES ROBERGE;YALEI LIU;ROBERT P. REHFUSS;CHARLES G. CLARK;PATRICK Y.S. LAM;ALEXANDRE L. L'HEUREUX;CARL THIBEAULT;GILLES BOUTHILLIER;DORA M. SCHNUR |
分类号 |
A61K31/444;A61K31/4439;A61K31/501;A61P7/02;C07C275/30;C07C275/32;C07D213/40;C07D213/75;C07D213/89;C07D231/40;C07D231/50;C07D237/22;C07D333/36;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07F7/18 |
主分类号 |
A61K31/444 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|