发明名称 N-SUBSTITUTED BENZIMIDAZOLYL C-KIT INHIBITORS AND COMBINATORIAL BENZIMIDAZOLE LIBRARY
摘要 Compounds represented by Formula (I) or a pharmaceutically acceptable salt or N-oxide thereof act as c-kit inhibitors and are useful in the treatment of tumors. Combinatorial libraries composed of compounds represented by Formula (I) or benzimidazole compounds represented by Formula (II) are useful in providing compounds to assay for such therapeutically useful compounds.
申请公布号 WO2006060381(A3) 申请公布日期 2006.12.28
申请号 WO2005US43114 申请日期 2005.11.30
申请人 OSI PHARMACEUTICALS, INC.;CREW, ANDREW, PHILIP;COX, MATTHEW;LAUFER, RADOSLAW;SUN, YINGCHUAN;PEGG, NEIL, ANTHONY;SAMBROOK SMITH, COLIN, PETER;WILKES, ROBIN, DAVID;WILLIAMS, JONATHAN 发明人 CREW, ANDREW, PHILIP;COX, MATTHEW;LAUFER, RADOSLAW;SUN, YINGCHUAN;PEGG, NEIL, ANTHONY;SAMBROOK SMITH, COLIN, PETER;WILKES, ROBIN, DAVID;WILLIAMS, JONATHAN
分类号 C07D235/06;A61K31/4184;A61P35/00;C07D401/12;C07D403/10;C07D403/14;C07D405/10;C07D409/10;C07D409/14;C07D413/10;C07D417/14;C40B40/04;C40B50/14 主分类号 C07D235/06
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