发明名称 |
Benzisothiazol-3-one-carboxylic acid amides as phospholipase inhibitors |
摘要 |
A novel class of benzisothiazole-3(2H)-one compounds is disclosed together with the use of such compounds for inhibiting hepatic lipase and/or endothelial lipase activity for treatment, amelioration or prevention of hepatic lipase and/or endothelial lipase mediated diseases. (I)
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申请公布号 |
US2006276522(A1) |
申请公布日期 |
2006.12.07 |
申请号 |
US20050550006 |
申请日期 |
2005.09.14 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
EACHO PATRICK I.;FOXWORTHY-MASON PATRICIA S.;LIN HO-SHEN;LOPEZ JOSE E.;MOSLOR MARIAN K.;RICHETT MICHAEL E. |
分类号 |
A61K31/425;A61P3/00;C07D275/04;C07D417/12 |
主分类号 |
A61K31/425 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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