发明名称 1, 6 -DIHYDRO- 1,3, 5, 6-TETRAAZA-AS-INDACENE BASED TRICYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME AS INHIBITORS OF IKK ENZYME ACTIVITY
摘要 <p>The present invention provides for tricyclic compounds having the formula (I) wherein R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;5&lt;/SUP&gt;, R&lt;SUP&gt;6&lt;/SUP&gt;, R&lt;SUP&gt;7&lt;/SUP&gt;, and R&lt;SUP&gt;8&lt;/SUP&gt; are as described herein. The present invention further provides pharmaceutical compositions comprising such compounds, as well as the use of such compounds for treating inflammatory and immune diseases.</p>
申请公布号 WO2006122137(A1) 申请公布日期 2006.11.16
申请号 WO2006US17950 申请日期 2006.05.09
申请人 BRISTOL-MYERS SQUIBB COMPANY;PITTS, WILLIAM J.;KEMPSON, JAMES;GUO, JUNQING;DAS, JAGABANDHU;LANGEVINE, CHARLES M.;SPERGEL, STEVEN H.;WATTERSON, SCOTT H. 发明人 PITTS, WILLIAM J.;KEMPSON, JAMES;GUO, JUNQING;DAS, JAGABANDHU;LANGEVINE, CHARLES M.;SPERGEL, STEVEN H.;WATTERSON, SCOTT H.
分类号 C07D471/14;A61K31/437;A61P11/06;A61P17/06;A61P19/02;A61P35/00 主分类号 C07D471/14
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