发明名称 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS
摘要 The present invention provides a pyrrolidine compound of General Formula (1) or a salt thereof, wherein R¿101? and R¿102? are each independently a phenyl group or a pyridyl group, the phenyl group or the pyridyl group may have one or more substituents selected from halogen atoms and lower alkyl groups optionally substituted with one or more halogen atoms, etc. The pyrrolidine compound or a salt thereof of the present invention is usable to produce a pharmaceutical preparation having a wider therapeutic spectrum and being capable of exhibiting sufficient therapeutic effects after short-term administration.
申请公布号 WO2006121218(A1) 申请公布日期 2006.11.16
申请号 WO2006JP309988 申请日期 2006.05.12
申请人 OTSUKA PHARMACEUTICAL CO., LTD.;KURIMURA, MUNEAKI;TAIRA, SHINICHI;TOMOYASU, TAKAHIRO;ITO, NOBUAKI;TAI, KUNINORI;TAKEMURA, NORIAKI;MATSUZAKI, TAKAYUKI;MENJO, YASUHIRO;MIYAMURA, SHIN;SAKURAI, YOHJI;WATANABE, AKIHITO;SAKATA, YASUYO;MASUMOTO, TAKUMI;AKAZAWA, KOHEI;SUGINO, HARUHIKO;AMADA, NAOKI;OHASHI, SATOSHI;SHINOHARA, TOMOICHI;SASAKI, HIROFUMI;MORITA, CHISAKO;YAMASHITA, JUNKO;NAKAJIMA, SATOKO 发明人 KURIMURA, MUNEAKI;TAIRA, SHINICHI;TOMOYASU, TAKAHIRO;ITO, NOBUAKI;TAI, KUNINORI;TAKEMURA, NORIAKI;MATSUZAKI, TAKAYUKI;MENJO, YASUHIRO;MIYAMURA, SHIN;SAKURAI, YOHJI;WATANABE, AKIHITO;SAKATA, YASUYO;MASUMOTO, TAKUMI;AKAZAWA, KOHEI;SUGINO, HARUHIKO;AMADA, NAOKI;OHASHI, SATOSHI;SHINOHARA, TOMOICHI;SASAKI, HIROFUMI;MORITA, CHISAKO;YAMASHITA, JUNKO;NAKAJIMA, SATOKO
分类号 C07D401/12;A61K31/40;A61K31/4439;A61K31/497;A61P25/00;C07D207/14;C07D401/14;C07D403/14;C07D405/12;C07D407/12;C07D407/14;C07D413/12;C07D413/14;C07D417/12;C07D417/14 主分类号 C07D401/12
代理机构 代理人
主权项
地址