发明名称 METHODS FOR PRODUCTION OF PEPTIDE DERIVATIVES
摘要 The invention relates to methods for the preparation of peptides which are a C-terminal amide derivatives by a combination of solid-phase synthesis and post assembly solution phase synthesis. The peptides which are a C-terminal amide derivatives are further converted to peptide acetates. The invention also relates to pure peptide acetates and to protected peptide precursors.
申请公布号 WO2006119388(A2) 申请公布日期 2006.11.09
申请号 WO2006US17044 申请日期 2006.05.02
申请人 NOVETIDE, LTD.;TEVA PHARMACEUTICALS USA, INC.;TOVI, AVI;EIDELMAN, CHAIM;SHUSHAN, SHIMON;ELSTER, SHAI;ALON, HAGI;IVCHENKO, ALEXANDER;BUTILCA, GABRIEL-MARCUS;ZAOVI, GIL;ALTERMAN, ELEONORA;BAR-OZ, LEAH;GADI, TEHILA 发明人 TOVI, AVI;EIDELMAN, CHAIM;SHUSHAN, SHIMON;ELSTER, SHAI;ALON, HAGI;IVCHENKO, ALEXANDER;BUTILCA, GABRIEL-MARCUS;ZAOVI, GIL;ALTERMAN, ELEONORA;BAR-OZ, LEAH;GADI, TEHILA
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