发明名称 4- (2, 6-DICHLOROBENZOYLAMINO) -lH-PYRAZOLE-3 -CARBOXYLIC ACID PIPERIDIN- 4 -YLAMID ACID ADDITION SALTS AS KINASE INHIBITORS
摘要 The invention provides an acid addition salt of 4-(2,6-dichloro-benzoylamino)-lH- pyrazole-3-carboxylic acid piperidin-4-ylamide and crystals thereof, the salt being formed with an acid selected from methanesulphonic acid and acetic acid and mixtures thereof. Also provided are the novel uses of salts of 4-(2,6-dichloro-benzoylamino)-lH- pyrazole-3-carboxylic acid piperidin-4-ylamide, processes for the preparation of 4- (2,6-dichloro-benzoylamino)-lH-pyrazole-3-carboxylic acid piperidin-4-ylamide and its salts and novel chemical intermediates.
申请公布号 WO2006077426(A3) 申请公布日期 2006.09.28
申请号 WO2006GB00207 申请日期 2006.01.20
申请人 ASTEX THERAPEUTICS LIMITED;WYATT, PAUL, GRAHAM;REES, DAVID, CHARLES;VINKOVIC, MLADEN;TREWARTHA, GARY 发明人 WYATT, PAUL, GRAHAM;REES, DAVID, CHARLES;VINKOVIC, MLADEN;TREWARTHA, GARY
分类号 C07D401/12;A61K31/4155;A61K31/454;A61P35/00;A61P35/02 主分类号 C07D401/12
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