发明名称 |
PROCESS AND METHODS FOR THE PREPARATION OF OPTICALLY ACTIVE CIS-2-HYDROXYMETHYL-4-(CYTOSIN-1´-YL)-1,3-OXATHIOLANE OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF |
摘要 |
<p>There is provided a method for resolving a compound of formula (III), in the cis configuration: There is also provided a process for producing optically active compound of formula (I) or (II): wherein: R<SUB>1</SUB>, R<SUB>2</SUB>, R<SUB>3</SUB> are as defined herein, the method and process involving the production, recovery and conversion of diastereomeric salts.</p> |
申请公布号 |
WO2006096954(A1) |
申请公布日期 |
2006.09.21 |
申请号 |
WO2005CA00384 |
申请日期 |
2005.03.14 |
申请人 |
SHIRE BIOCHEM INC.;CIMPOIA, ALEX |
发明人 |
CIMPOIA, ALEX;SIMION, DAN |
分类号 |
C07D411/04 |
主分类号 |
C07D411/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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