发明名称 PRODRUG CONSTRUCTS OF PYRIMIDINONE COMPOUNDS AS CALCILYTICS
摘要 Various calcilytic compounds and prodrugs of calcilytic compounds are disclosed. Calcilytic compounds are compounds capable of inhibiting calcium receptor activity. Methods for preparing these compounds, oral bioavailability of these compounds, pharmaceutical compositions containing these compounds and their use as calcium receptor antagonists are also disclosed.
申请公布号 WO2006066070(A3) 申请公布日期 2006.09.21
申请号 WO2005US45565 申请日期 2005.12.16
申请人 NPS PHARMACEUTICALS, INC.;SHCHERBAKOVA, IRINA;WERMUTH, CAMILLE, G.;JEANNOT, FREDERIC;CIAPETTI, PAOLA;ROQUES, VIRGINIE;JUNG, LAETITIA, M.;BALANDRIN, MANUEL, F.;NAIR, SATHEESH, K.;SWIERCZEK, KRZYSZTOF;MCCAFFREY, JENNIFER;HEATON, WILLIAM, L.;BREINHOLT, JEFF, A.;CONKLIN, REBECCA, L. 发明人 SHCHERBAKOVA, IRINA;WERMUTH, CAMILLE, G.;JEANNOT, FREDERIC;CIAPETTI, PAOLA;ROQUES, VIRGINIE;JUNG, LAETITIA, M.;BALANDRIN, MANUEL, F.;NAIR, SATHEESH, K.;SWIERCZEK, KRZYSZTOF;MCCAFFREY, JENNIFER;HEATON, WILLIAM, L.;BREINHOLT, JEFF, A.;CONKLIN, REBECCA, L.
分类号 C07D239/36;A61K31/513;C07C229/12 主分类号 C07D239/36
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