发明名称 BENZOXAZINONE DOPAMINE D4 RECEPTOR ANTAGONIST
摘要 <p>The invention relates to compounds having formulae (I) and (II) wherein R1 and R2 are independently hydrogen or C1-C6 alkyl; X is N or CH; and R3 is phenyl, naphtyl, heteroaryl, substituted phenyl, substituted naphtyl, or substituted heteroaryl, wherein each substituent is independently selected from halogen, C1-C6 alkoxy, C1-C6 alkyl, -CN, -CF3 or sulphonamido and pharmaceutically acceptable salts, esters, amides prodrugs thereof, that are antagonists of dopamine D4 receptor.</p>
申请公布号 RO120845(B1) 申请公布日期 2006.08.30
申请号 RO19980001622 申请日期 1997.05.20
申请人 WARNER-LAMBERT COMPANY 发明人 BELLIOTTI THOMAS;WISE LAWRENCE DAVID;WUSTROW DAVID JUERGEN
分类号 C07D265/36;A61K31/00;A61K31/535;A61K31/5375;A61K31/5377;A61P25/18;C07D413/06;C07D413/12;C07D417/12 主分类号 C07D265/36
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