摘要 |
A COMPOUND OF THE FORMULA FORMULA WHEREIN R1, R2 AND R3 ARE AS DEFINED ABOVE, WHICH ARE INHIBITORS OF THE ENZYME PROTEIN TYROSINE KINASES SUCH AS JANUS KINASE 3 AND AS SUCH ARE USEFUL THERAPY AS IMMUNOSUPPRESSIVE AGENTS FOR ORGAN TRANSPLANTS, LUPUS, MULTIPLE SCLEROSIS, RHEUMATOID, ARTHRITIS, PSORIASIS, TYPE I DIABETES AND COMPLICATIONS FROM DIABETES, CANCER, ASTHMA, ATOPIC DERMATITIS, AUTOIMMUNE THYROID DISORDERS, ULCERATIVE COLITIS, CROHN'S DISEASE, ALZHEIMER'S DISEASE, LEUKEMIA AND OTHER AUTOIMMUNE DISEASES.
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