发明名称 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF HISTONE DEACETYLASE
摘要 <p>Disclosed are compounds of formula (I) that inhibit histone deacetylase (HDAC) enzymatic activity, pharmaceutical compositions comprising such compounds, as well as methods to treat conditions, particularly proliferative conditions, mediated at least in part by HDAC, wherein A, W, W&lt;SUP&gt;1&lt;/SUP&gt;, W&lt;SUP&gt;2&lt;/SUP&gt;, Ar&lt;SUP&gt;2&lt;/SUP&gt;, and G are described herein.</p>
申请公布号 WO2006088949(A1) 申请公布日期 2006.08.24
申请号 WO2006US05312 申请日期 2006.02.14
申请人 MIKANA THERAPEUTICS, INC.;ANANDAN, SAMPATH, K.;XIAO, XIAO-YI;WARD, JOHN, S.;PATEL, DINESH, V. 发明人 ANANDAN, SAMPATH, K.;XIAO, XIAO-YI;WARD, JOHN, S.;PATEL, DINESH, V.
分类号 C07D471/04;A61K31/4353;A61P35/00;C07D401/04;C07D487/04;C07D491/04;C07D495/04 主分类号 C07D471/04
代理机构 代理人
主权项
地址