发明名称 Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substitutent in the 4-or 4'-position
摘要 What is described are a compound of the formula (I): wherein n is 0 or 1; A-B is -CH-CH- or -CH<SUB>2</SUB>-CH<SUB>2</SUB>-; R<SUB>1 </SUB>is C<SUB>1</SUB>-C<SUB>12</SUB>-alkyl, C<SUB>3</SUB>-C<SUB>8</SUB>-cycloalkyl or C<SUB>2</SUB>-C<SUB>12</SUB>-alkenyl; R<SUB>2 </SUB>is for example C<SUB>1</SUB>-C<SUB>12</SUB>-alkyl, C<SUB>2</SUB>-C<SUB>12</SUB>-alkenyl or C<SUB>2</SUB>-C<SUB>12</SUB>-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, -N<SUB>3</SUB>, -N0<SUB>2</SUB>, C<SUB>3</SUB>-C<SUB>8</SUB>-Cycloalkyl, norbornylenyl-, C<SUB>3</SUB>-C<SUB>8</SUB>Cycloalkenyl; C<SUB>3</SUB>-C<SUB>8</SUB>-halocycloalkyl, C<SUB>1</SUB>-C<SUB>12</SUB>-alkoxy, C<SUB>1</SUB>-C<SUB>6</SUB>-alkoxy-C<SUB>1</SUB>-C<SUB>6</SUB>-alkoxy, C<SUB>3</SUB>-C<SUB>8</SUB>-cycloalkoxy, C<SUB>1</SUB>-C<SUB>12</SUB>-haloalkoxy, C<SUB>1</SUB>-C<SUB>12</SUB>-alkylthio, C<SUB>3</SUB>-C<SUB>8</SUB>-cycloalkylthio, C<SUB>1</SUB>-C<SUB>12</SUB>-haloalkylthio, C<SUB>1</SUB>-C<SUB>12 </SUB>alkylsulfinyl, C<SUB>3</SUB>-C<SUB>8</SUB>-cycloalkylsulfinyl, C<SUB>1</SUB>-C<SUB>12</SUB>-haloalkylsulfinyl, C<SUB>3</SUB>-C<SUB>8</SUB>-halocycloalkylsulfinyl, C<SUB>1</SUB>-C<SUB>12</SUB>-alkylsulfonyl, C<SUB>3</SUB>-C<SUB>8</SUB>-cycloalkylsulfonyl, C<SUB>1</SUB>-C<SUB>12</SUB>haloalkylsulfonyl, C<SUB>3</SUB>-C<SUB>8</SUB>-halocycloalkylsulfonyl, -NR<SUB>4</SUB>R<SUB>6</SUB>, -X-C(-Y)-R<SUB>4</SUB>, -X-C(-Y)-Z-R<SUB>4</SUB>, -P(-O)(OC<SUB>1</SUB>-C<SUB>6</SUB>-alkyl)<SUB>2</SUB>, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R<SUB>3 </SUB>is for example H, C<SUB>1</SUB>-C<SUB>12</SUB>-alkyl or C<SUB>1</SUB>-C<SUB>12</SUB>-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
申请公布号 US2006148729(A1) 申请公布日期 2006.07.06
申请号 US20030539274 申请日期 2003.12.19
申请人 MAIENFISCH PETER;KESSABI FIONA M;CASSAYRE JEROME;QUARANTA LAURA;PITTERNA THOMAS;HUETER OTTMAR F;JUNG PIERRE 发明人 MAIENFISCH PETER;KESSABI FIONA M.;CASSAYRE JEROME;QUARANTA LAURA;PITTERNA THOMAS;HUETER OTTMAR F.;JUNG PIERRE
分类号 A01N43/04;A61K31/70;A61P33/00;C07H17/08 主分类号 A01N43/04
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