发明名称 |
Substituted alpha-halo-beta-keto-pyridinylpropanoates |
摘要 |
<p>The invention relates to 3-ketoester of formula (IV)
<Chemistry id="chema01" num="0001"><Image id="ia01" he="27" wi="52" file="IMGA0001.TIF" imgContent="chem" imgFormat="TIFF" /></Chemistry>
wherein R1 represents a 2, 3 or 4-pyridine ring optionally substituted by a C<Sub>3-6</Sub> cycloalkyl group, a C<Sub>1-4</Sub> alkyl group, a C<Sub>1-4</Sub> alkoxy group, a benzyl group or a halogen atom, R5 is an halogen atom and R is an alkyl.</p> |
申请公布号 |
EP1674456(A3) |
申请公布日期 |
2006.07.05 |
申请号 |
EP20050016160 |
申请日期 |
2002.09.19 |
申请人 |
SANOFI-AVENTIS;MITSUBISHI PHARMA CORPORATION |
发明人 |
GALLET, THIERRY;LARDENOIS, PATRICK;LOCHEAD, ALISTAIR;MARGUERIE, SEVERINE;NEDELEC, ALAIN;SAADY, MOURAD;SLOWINSKI, FRANCK;YAICHE, PHILIPPE |
分类号 |
C07D213/60;A61K31/519;A61P3/04;A61P3/10;A61P9/10;A61P17/14;A61P25/00;A61P25/02;A61P25/08;A61P25/16;A61P25/18;A61P25/24;A61P25/28;A61P27/02;A61P27/06;A61P35/00;A61P43/00;C07D213/50;C07D487/04 |
主分类号 |
C07D213/60 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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