发明名称 Avermectin and avermectin monosaccharide derivatives substituted in the 4-or 4'-position having pesticidal properties
摘要 What is described are a compound of the formula (I) Wherein U is -N(R<SUB>2</SUB>)OR<SUB>3 </SUB>or -N<SUP>+</SUP>(O<SUP>-</SUP>)-C(R<SUB>E</SUB>)R<SUB>Z</SUB>); n is 0 or 1; X-Y is -CH-CH- or -CH<SUB>2</SUB>-CH<SUB>2</SUB>-; R<SUB>1 </SUB>is C<SUB>1</SUB>-C<SUB>12</SUB>alkyl, C<SUB>3</SUB>-C<SUB>8</SUB>cycloalkyl or C<SUB>2</SUB>-C<SUB>12</SUB>alkenyl; R<SUB>2 </SUB>and R<SUB>3 </SUB>are, for example; independently from each other, -Q, -C(-O)-Z-Q or -CN; R<SUB>Z </SUB>and R<SUB>E </SUB>are, independently from each other, -Q, -C(-O)-Z-Q or -CN; or R<SUB>Z </SUB>and R<SUB>E </SUB>together are a three- to seven membered alkylene or alkenylene bridge, which is unsubstituted or mono- to tri-substituted; Z is a bond, O or -NR<SUB>4</SUB>-; Q is H, C<SUB>1</SUB>-C<SUB>12</SUB>alkyl, C<SUB>2</SUB>-C<SUB>12</SUB>alkenyl, C<SUB>2</SUB>-C<SUB>12</SUB>alkynyl, C<SUB>3</SUB>-C<SUB>12</SUB>-Cycloalkyl, C<SUB>5</SUB>-C<SUB>12</SUB>-cycloalkenyl, aryl, or heterocyclyl, which are unsubstituted or mono- to pentasubstituted; R<SUB>4 </SUB>is for example H, C<SUB>1</SUB>-C<SUB>8</SUB>alkyl, hydroxy-C<SUB>1</SUB>-C<SUB>8</SUB>alkyl, C<SUB>3</SUB>-C<SUB>8</SUB>cycloalkyl or C<SUB>2</SUB>-C<SUB>8</SUB>alkenyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.
申请公布号 US2006140997(A1) 申请公布日期 2006.06.29
申请号 US20050543637 申请日期 2005.07.28
申请人 PITTERNA THOMAS;KESSABI FIONA M;MAIENFISCH PETER;CASSAYRE JEROME;JUNG PIERRE;QUARANTA LAURA 发明人 PITTERNA THOMAS;KESSABI FIONA M.;MAIENFISCH PETER;CASSAYRE JEROME;JUNG PIERRE;QUARANTA LAURA
分类号 A01N25/00;A01N43/04;A61P33/00;C07H17/08 主分类号 A01N25/00
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