发明名称 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE)
摘要 The present invention is directed to novel 2-amino-3, 4-dihydro­quinazoline derivatives, pharmaceutical compositions containing them and their use in the treatment of Alzheimer's disease (AD) and related disorders. The compounds of the invention are inhibitors of P-secretase, also known as n-site cleaving enzyme and BACE.
申请公布号 WO2006017836(A3) 申请公布日期 2006.06.29
申请号 WO2005US28191 申请日期 2005.08.08
申请人 JANSSEN PHARMACEUTICA, N.V.;BAXTER, ELLEN;BISCHOFF, FRANCOIS, PAUL;BOYD, ROBERT;BRAEKEN, MIRIELLE;COATS, STEVEN;HUANG, YIFANG;JORDAN, ALFONZO;LUO, CHI;MERCKEN, MARC, HUBERT;REYNOLDS, CHARLES, H.;ROSS, TINA, MORGAN;TOUNGE, BRETT, A.;SCHULZ, MARK;DE WINTER, HANS, LOUIS, JOS;PIETERS, SERGE MARIA ALOYSIUS;REITZ, ALLEN, B. 发明人 BAXTER, ELLEN;BISCHOFF, FRANCOIS, PAUL;BOYD, ROBERT;BRAEKEN, MIRIELLE;COATS, STEVEN;HUANG, YIFANG;JORDAN, ALFONZO;LUO, CHI;MERCKEN, MARC, HUBERT;REYNOLDS, CHARLES, H.;ROSS, TINA, MORGAN;TOUNGE, BRETT, A.;SCHULZ, MARK;DE WINTER, HANS, LOUIS, JOS;PIETERS, SERGE MARIA ALOYSIUS;REITZ, ALLEN, B.
分类号 C07D239/84;A61K31/517;A61P25/28 主分类号 C07D239/84
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