发明名称 |
DEPRESSION OF HERG K+ CHANNEL FUNCTION IN MAMMALIAN CELLS AND APPLICATIONS TO THE CONTROL OF CANCER CELLS DIVISION |
摘要 |
<p>The use of an HERG channel inhibitor for controlling the proliferation of cancer cells. Examples of such HERG channel inhibitors include dofetilide, cisapride, E-4031 and a siRNA molecule targeting a sequence involved in the expression of an HERG channel. Other ERG channels are also targets for these inhibitors.</p> |
申请公布号 |
WO2006039806(A1) |
申请公布日期 |
2006.04.20 |
申请号 |
WO2005CA01574 |
申请日期 |
2005.10.14 |
申请人 |
INSTITUT DE CARDIOLOGIE DE MONTREAL;YANG, BAOFENG;WANG, ZHIGUO |
发明人 |
WANG, ZHIGUO |
分类号 |
A61K31/4545;C07H21/02;A61K31/18;A61K31/4468;A61K31/7105;A61K48/00;A61P35/00 |
主分类号 |
A61K31/4545 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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