发明名称 USE OF PURIFIED DONEPEZIL MALEATE FOR PREPARING PHARMACEUTICALLY PURE AMORPHOUS DONEPEZIL HYDROCHLORIDE
摘要 <p>The present invention provides a crystalline donepezil maleate, which is used as an intermediate in the preparation of donepezil hydrochloride. Also provided are novel processes for producing same in substantially pure form and a process for producing pharmaceutically pure amorphous donepezil hydrochloride therefrom.</p>
申请公布号 WO2006035433(A2) 申请公布日期 2006.04.06
申请号 WO2005IL01034 申请日期 2005.09.27
申请人 CHEMAGIS LTD.;ARAD, ODED;ZELIKOVITCH, LIOR;ALNABARI, MOHAMMED;BRAND, MICHAEL;GRIBUN, IRINA;SALMAN, ADA;SHIFFER, MEITAL;SHOOKRUN, MOTY;KURLAT, ORNA;BENTOLILA, MOSHE;KASPI, JOSEPH 发明人 ARAD, ODED;ZELIKOVITCH, LIOR;ALNABARI, MOHAMMED;BRAND, MICHAEL;GRIBUN, IRINA;SALMAN, ADA;SHIFFER, MEITAL;SHOOKRUN, MOTY;KURLAT, ORNA;BENTOLILA, MOSHE;KASPI, JOSEPH
分类号 A61K31/445;C07D211/06 主分类号 A61K31/445
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