发明名称 |
HETEROCYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS |
摘要 |
Methods of treating an SCD-mediated disease or condition in a mammal, preferably a human, are disclosed, wherein the methods comprise administering to a mammal in need thereof a compound of formula (I): where x, y, G, J, K, L, M, V R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, R<SUP>5a</SUP>, R<SUP>6</SUP>, R<SUP>6a</SUP>, R<SUP>7</SUP>, R<SUP>7a</SUP>, R<SUP>8</SUP> and R<SUP>8a</SUP> are defined herein. Pharmaceutical compositions comprising the compounds of formula (I) are also disclosed. |
申请公布号 |
WO2006034440(A2) |
申请公布日期 |
2006.03.30 |
申请号 |
WO2005US34129 |
申请日期 |
2005.09.20 |
申请人 |
XENON PHARMACEUTICALS INC.;KAMBOJ, RAJENDER;ZHANG, ZAIHUI;FU, JIAN-MIN;KODUMURU, VISHNUMURTHY;SVIRIDOV, SERGUEI;SADALAPURE, KASHINATH;LIU, SHIFENG;SUN, SHAOYI;HOU, DUANJIE;CHAKKA, NAGASREE |
发明人 |
KAMBOJ, RAJENDER;ZHANG, ZAIHUI;FU, JIAN-MIN;KODUMURU, VISHNUMURTHY;SVIRIDOV, SERGUEI;SADALAPURE, KASHINATH;LIU, SHIFENG;SUN, SHAOYI;HOU, DUANJIE;CHAKKA, NAGASREE |
分类号 |
A61K31/501;A61K31/496;A61P1/16;A61P3/00;A61P3/04;A61P3/06;A61P3/10;C07D403/00 |
主分类号 |
A61K31/501 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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