发明名称 METHANESULFONIC ACID SALT OF PYRAZOLOPYRIMIDINE COMPOUND, CRYSTAL THEREOF, AND PROCESS FOR PRODUCING THE SAME.
摘要 <p>8-(3-Pentylamino)-2-methyl-3-(2-chloro-4-methoxy -phenyl)-6,7-dihydro-5H-cyclopenta[d]pyrazolo[1,5-a] -pyrimidine methanesulfonate, which is novel, and a process for producing an intermediate for the compound. 8-(3-Pentylamino)-2-methyl-3-(2-chloro-4-methoxy -phenyl)-6,7-dihydro-5H-cyclopenta[d]pyrazolo[1,5-a] -pyrimidine methanesulfonate is a compound having highly excellent thermal stability. The novel production process enables a compound represented by the general formula (I): (I) (wherein Ar represents an optionally substituted benzene ring, etc.; and R1 represents C1-8 alkyl, C2-8 alkenyl, C2-8 alkynyl, etc.), which is an intermediate, to be efficiently produced in a high yield.</p>
申请公布号 MXPA05013917(A) 申请公布日期 2006.03.09
申请号 MX2005PA13917 申请日期 2004.06.24
申请人 ONO PHARMACEUTICAL CO., LTD. 发明人 MASAKI OKAMOTO
分类号 A61K31/519;A61K9/08;A61K47/10;A61P1/00;A61P5/04;A61P5/10;A61P15/00;A61P25/00;A61P29/00;A61P37/00;C07C253/30;C07C255/40;C07D487/04;(IPC1-7):A61K31/519 主分类号 A61K31/519
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