发明名称 A NOVEL POLYMORPH OF (1-BENZYL-4-[(5,6-DIMETHOXY-1-INDANONE)-2-YL] METHYL PIPERIDINE HYDROCHLORIDE (DONEPEZIL HYDROCHLORIDE) AND A PROCESS FOR PRODUCING THEREOF
摘要 <p>The present invention discloses a novel, stable polymorph of 1-benzyl-4-[(5,6 dimethoxy-l-indanone)-2-y1] methyl piperidine hydrochloride commonly known as Donepezil hydrochloride. Further the present invention discloses a process for producing Donepezil HCl amorphous and it's polymorph Form (VI).</p>
申请公布号 WO2006011154(A1) 申请公布日期 2006.02.02
申请号 WO2004IN00227 申请日期 2004.07.28
申请人 USV LIMITED;TARUR, VENKATASUBRAMANIAN, RADHAKRISHNAN;SATHE, DHANANJAY, GOVIND;NAIDU, AVINASH, VENKATARAMAN;AHER, UMESH, PARASHRAM;SAWANT, KAMLESH, DIGAMBAR 发明人 TARUR, VENKATASUBRAMANIAN, RADHAKRISHNAN;SATHE, DHANANJAY, GOVIND;NAIDU, AVINASH, VENKATARAMAN;AHER, UMESH, PARASHRAM;SAWANT, KAMLESH, DIGAMBAR
分类号 C07D211/32;(IPC1-7):C07D211/32;A61P25/28;A61K31/445 主分类号 C07D211/32
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