发明名称 АМИДЫ АМИНОАЛКИЛЗАМЕЩЕННЫХ АЗЕТИДИНОВ, ПИРРОЛИДИНОВ, ПИПЕРИДИНОВ И АЗЕПАНОВ
摘要 Novel amides of aminoalkyl-substituted azetidines, pyrrolidines, piperidines and azepanes, use of these compounds as pharmaceutical compositions, pharmaceutical compositions comprising the compounds, and a method of treatment employing these compounds and compositions. The compounds show a high and selective binding affinity to the histamine H3 receptor indicating histamine H3 receptor antagonistic, inverse agonistic or agonistic activity. As a result, the compounds are useful for the treatment of diseases and disorders related to the histamine H3 receptor.
申请公布号 RU2004126438(A) 申请公布日期 2006.01.27
申请号 RU20040126438 申请日期 2003.01.27
申请人 НОВО НОРДИСК А/С (DK) 发明人 ПЕШКЕ Бернд (DK);ПЕТТЕРССОН Ингрид (DK)
分类号 C07D403/06;A61K31/4025;A61K31/4196;A61K31/454;A61P1/04;A61P1/08;A61P1/12;A61P1/16;A61P3/00;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P9/12;A61P11/02;A61P11/06;A61P19/02;A61P25/00;A61P25/06;A61P25/08;A61P25/20;A61P25/24;A61P25/26;A61P25/28;A61P35/00;A61P37/00;A61P37/08;A61P43/00;C07D207/09;C07D211/26;C07D403/10;C07D405/06;C07D409/06;C07D521/00 主分类号 C07D403/06
代理机构 代理人
主权项
地址