发明名称 |
АМИДЫ АМИНОАЛКИЛЗАМЕЩЕННЫХ АЗЕТИДИНОВ, ПИРРОЛИДИНОВ, ПИПЕРИДИНОВ И АЗЕПАНОВ |
摘要 |
Novel amides of aminoalkyl-substituted azetidines, pyrrolidines, piperidines and azepanes, use of these compounds as pharmaceutical compositions, pharmaceutical compositions comprising the compounds, and a method of treatment employing these compounds and compositions. The compounds show a high and selective binding affinity to the histamine H3 receptor indicating histamine H3 receptor antagonistic, inverse agonistic or agonistic activity. As a result, the compounds are useful for the treatment of diseases and disorders related to the histamine H3 receptor. |
申请公布号 |
RU2004126438(A) |
申请公布日期 |
2006.01.27 |
申请号 |
RU20040126438 |
申请日期 |
2003.01.27 |
申请人 |
НОВО НОРДИСК А/С (DK) |
发明人 |
ПЕШКЕ Бернд (DK);ПЕТТЕРССОН Ингрид (DK) |
分类号 |
C07D403/06;A61K31/4025;A61K31/4196;A61K31/454;A61P1/04;A61P1/08;A61P1/12;A61P1/16;A61P3/00;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P9/12;A61P11/02;A61P11/06;A61P19/02;A61P25/00;A61P25/06;A61P25/08;A61P25/20;A61P25/24;A61P25/26;A61P25/28;A61P35/00;A61P37/00;A61P37/08;A61P43/00;C07D207/09;C07D211/26;C07D403/10;C07D405/06;C07D409/06;C07D521/00 |
主分类号 |
C07D403/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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