发明名称 |
AZETIDINECARBOXAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CB1 RECEPTOR MEDIATED DISORDERS. |
摘要 |
<p>Compounds of formula (I) and their use in therapy, particularly for the treatment of a disorder mediated by CB1 receptors such as obesity: Formuila (I) wherein: R1 and R2 are independently selected from aryl; and R3 is hydrogen or alkyl; or a pharmaceutically acceptable salt or prodrug thereof, wherein at least one of R1 and R2 has a non-hydrogen substituent in the ortho-position(s) thereof relative to the point of attachment to the [-CH-0-] group.</p> |
申请公布号 |
MXPA05011670(A) |
申请公布日期 |
2005.12.15 |
申请号 |
MX2005PA11670 |
申请日期 |
2004.04.29 |
申请人 |
VERNALIS RESEARCH LIMITED. |
发明人 |
SUKHJIT SOHAL |
分类号 |
A61P3/04;C07D205/04;C07D405/12;C07D409/12;(IPC1-7):A61K31/397;C07D413/12 |
主分类号 |
A61P3/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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