发明名称 |
4- 2- (CYCLOALKYLAMINO) PYRIMIDIN-4-YL ! - (PHENYL) - IMIDAZOLIN-2- ONE DERIVATIVES AS P38 MAP- KINASE INHIBITORS FOR THE TREATMENT OF INFLAMMATORY DISEASES |
摘要 |
<p>The present invention is to provide a novel heterocyclic compound of the formula [I]: wherein R¿1< is a halogen, nitro, an alkyl, etc.; R¿2? is hydrogen, an alkyl, etc.; Ring A is 2-oxo-4-imidazolin-3,4-diyl, etc.; Ring B is a cycloalkyl, monocyclic saturated heterocyclic group; X is CH, N; Y is a single bond, CO, SO2; Z is O, NH, etc.; and Ring C is an aryl, a heterocyclic group, or a pharmaceutically acceptable salt thereof, which is useful as a p38 MAP kinase inhibitor.</p> |
申请公布号 |
WO2005105790(A1) |
申请公布日期 |
2005.11.10 |
申请号 |
WO2005JP08564 |
申请日期 |
2005.04.28 |
申请人 |
TANABE SEIYAKU CO., LTD.;KUBO, AKIRA;NAKANE, TETSU;NAKAJIMA, TATSUO;MURAKAMI, TAKANORI;MIYOSHI, HIDETAKA;OGASAWARA, AKIHITO |
发明人 |
KUBO, AKIRA;NAKANE, TETSU;NAKAJIMA, TATSUO;MURAKAMI, TAKANORI;MIYOSHI, HIDETAKA;OGASAWARA, AKIHITO |
分类号 |
A61K31/506;C07D401/14;C07D403/04;C07D403/14;C07D405/14;C07D409/14;C07D413/14;C07D417/14;(IPC1-7):C07D403/14;A61P29/00 |
主分类号 |
A61K31/506 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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