发明名称 PROCESS FOR THE PREPARATION OF PERINDOPRIL
摘要 <p>A process for preparing perindopril (III) or a pharmaceutically acceptable salt thereof, which process comprises a substituted benzyl ester of (2S,3aS,7aS)-octahydroindole-2-carboxylic acid (I) with N-[(S)-carbethoxybutyl]-(S)-alanine (II) where R represents a halo, C1-4 alkoxy or nitro substituent.</p>
申请公布号 WO2005100317(A1) 申请公布日期 2005.10.27
申请号 WO2005GB01355 申请日期 2005.04.07
申请人 NEOPHARMA LIMITED;NEOPHARMA LIMITED;KANKAN, RAJENDRA, NARAYANRAO;RAO, DHARMARAJ, RAMACHANDRA;WAIN, CHRISTOPHER, PAUL 发明人 KANKAN, RAJENDRA, NARAYANRAO;RAO, DHARMARAJ, RAMACHANDRA
分类号 C07D209/42;C07K5/06;(IPC1-7):C07D209/42 主分类号 C07D209/42
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