<p>A process for preparing perindopril (III) or a pharmaceutically acceptable salt thereof, which process comprises a substituted benzyl ester of (2S,3aS,7aS)-octahydroindole-2-carboxylic acid (I) with N-[(S)-carbethoxybutyl]-(S)-alanine (II) where R represents a halo, C1-4 alkoxy or nitro substituent.</p>
申请公布号
WO2005100317(A1)
申请公布日期
2005.10.27
申请号
WO2005GB01355
申请日期
2005.04.07
申请人
NEOPHARMA LIMITED;NEOPHARMA LIMITED;KANKAN, RAJENDRA, NARAYANRAO;RAO, DHARMARAJ, RAMACHANDRA;WAIN, CHRISTOPHER, PAUL