发明名称 |
Substituted pyrazolyl compounds for the treatment of inflammation |
摘要 |
The present invention relates to substituted pyrazolyl derivatives, compositions comprising such, intermediates, methods of making substituted pyrazolyl derivatives, and methods for treating cancer, inflammation, and inflammation-associated disorders, such as arthritis.
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申请公布号 |
US6956052(B2) |
申请公布日期 |
2005.10.18 |
申请号 |
US20020247096 |
申请日期 |
2002.09.19 |
申请人 |
PHARMACIA CORPORATION |
发明人 |
BERGMANIS ARIJA A.;CLARE MICHAEL;CRICH JOYCE Z.;GENG LIFENG;HAGEN TIMOTHY J.;HANSON GUNNAR J.;HOUDEK STEPHEN C.;HUANG HE;IULA DONNA M.;KOSZYK FRANCIS J.;LIAO SHUYUAN;MOHLER SCOTT B.;NGUYEN MARIA;PARTIS RICHARD A.;STEALEY MICHAEL A.;TOLLEFSON MICHAEL B.;WEIER RICHARD M.;XU XIANGDONG;BONAFOUX DOMINIQUE;FLETCHER THERESA R.;HAMPER BRUCE C.;LENNON PATRICK J.;LIAO SUBO;METZ SUZANNE;OBURN DAVID S.;OWEN THOMAS J.;SCATES ANGELA M.;VAZQUEZ MICHAEL L.;WOLFSON SERGE G. |
分类号 |
A61K31/416;A61K31/4178;A61K31/4245;A61K31/427;A61K31/433;A61K31/437;A61K31/4439;A61K31/444;A61K31/4709;A61K31/4725;A61K31/496;A61K31/506;A61K31/5377;A61K31/551;A61P19/02;A61P25/04;A61P29/00;A61P35/00;C07D231/54;C07D333/62;C07D401/04;C07D401/10;C07D401/12;C07D401/14;C07D403/12;C07D405/04;C07D405/10;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07D417/14;C07D471/04;(IPC1-7):A61K31/416 |
主分类号 |
A61K31/416 |
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