发明名称 |
4-(2-KETO-1-BENZIMIDAZOLINYL)PIPERIDINE COMPOUNDS AS ORL1-RECEPTOR AGONISTS |
摘要 |
A compound of formula (I) or the pharmaceutically acceptable salts thereof, wherein R1, R2, R3, R4 and R5 are defined above are useful as ORL1-receptor agonists, and useful as analgesics or the like in mammalian subjects. |
申请公布号 |
CA2317462(C) |
申请公布日期 |
2005.09.13 |
申请号 |
CA19992317462 |
申请日期 |
1999.01.08 |
申请人 |
PFIZER LIMITED |
发明人 |
KONDO, HIROSHI;NOGUCHI, HIROHIDE;OHASHI, YORIKO;YAMAGISHI, TATSUYA;ITO, FUMITAKA |
分类号 |
A61K31/4427;A61K31/4433;A61K31/454;A61K31/4545;A61K31/496;A61K31/506;A61K31/5377;A61P7/12;A61P9/12;A61P23/00;A61P25/04;A61P25/22;A61P29/00;A61P43/00;C07D401/04;C07D401/14;C07D409/14;(IPC1-7):C07D401/04;A61K31/445 |
主分类号 |
A61K31/4427 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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