发明名称 ACYLATED PIPERIDINE DERIVATIVES AS MELANOCORTIN-4 RECEPTOR AGONITS
摘要 Certain novel 4-substituted N-acylated piperidine derivatives are agonists of the human melanocortin receptor(s) and, in particular, are selective agonists of the human melanocortin-4 receptor (MC-4R). They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the activation of MC-4R, such as obesity, diabetes, sexual dysfunction, including erectile dysfunction and female sexual dysfunction.
申请公布号 HRP20030668(A2) 申请公布日期 2005.08.31
申请号 HR2003P000668 申请日期 2003.08.22
申请人 MERCK & CO. INC. 发明人 FEROZE UJJAINWALLA;LIN CHU;MARK T. GOULET;BONNIE LOURIDAS;DANIEL WARNER;MATTHEW J. WYVRATT
分类号 A61K31/445;A61K31/454;A61K31/504;A61K31/505;A61K31/5377;A61K45/00;A61P3/04;A61P3/06;A61P3/10;A61P9/12;A61P15/10;A61P17/10;A61P19/02;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P29/00;A61P35/00;A61P37/00;A61P43/00;C07D211/62;C07D211/64;C07D401/06;C07D401/14;C07D413/06;C07D413/14;C07D417/14;C07D451/02;C07D491/08 主分类号 A61K31/445
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