发明名称 IMIDAZOPYRIDIN-DERIVATE
摘要 The present invention relates to novel compounds having a phosphatidylinositol 3 kinase (PI3K) inhibiting activity which are useful as medicaments, more particularly as antitumor agent. Novel 3-(imidazoÄ1,2-aÜpyridin-3-yl) derivatives or salts thereof exhibit an excellent PI3K inhibiting activity and cancer cell growth inhibiting activity, and are thus useful as medicaments, especially as PI3K inhibitors and antitumor agents.
申请公布号 AT300540(T) 申请公布日期 2005.08.15
申请号 AT20010925980T 申请日期 2001.04.26
申请人 YAMANOUCHI PHARMACEUTICAL CO. LTD.;LUDWIG INSTITUTE FOR CANCER RESEARCH;IMPERIAL CANCER RESEARCH TECHNOLOGY LIMITED 发明人 HAYAKAWA, MASAHIKO;KAIZAWA, HIROYUKI;KAWAGUCHI, KEN-ICHI;MATSUDA, KOYO;ISHIKAWA, NORIKO;KOIZUMI, TOMONOBU;YAMANO, MAYUMI;OKADA, MINORU;OHTA, MITSUAKI
分类号 A61P35/00;A61P43/00;C07D471/04;C07D487/04;(IPC1-7):C07D471/04;A61K31/437;A61K31/470;A61K31/454;A61K31/537;A61K31/496;A61K31/444 主分类号 A61P35/00
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