发明名称 |
НОВЫЙ КРИСТАЛЛ ПРОИЗВОДНОГО АРИЛЭТЕНСУЛЬФОНАМИДА И СПОСОБ ЕГО ПОЛУЧЕНИЯ |
摘要 |
Crystalline (E)-N-[(6-methoxy-5-(2-methoxyphenoxy)-2-pyrimidin-2-yl)pyrimidin-4-yl]-2-phenylethenesulfonamide (I) potassium salt is new. Crystalline (E)-N-[(6-methoxy-5-(2-methoxyphenoxy)-2-pyrimidin-2-yl)pyrimidin-4-yl]-2-phenylethenesulfonamide of formula (I) potassium salt is new. [Image] An independent claim is included for the solvates of (I) with ethyl acetate and ethanol. ACTIVITY : Cardiovascular-Gen.; Hypotensive. MECHANISM OF ACTION : Endothelin-Agonist-A; Endothelin-Antagonist-A. |
申请公布号 |
RU2004105867(A) |
申请公布日期 |
2005.06.27 |
申请号 |
RU20040105867 |
申请日期 |
2002.07.25 |
申请人 |
ЯМАНОУТИ ФАРМАСЬЮТИКАЛ КО.,ЛТД. (JP) |
发明人 |
КАТО Ёсинори (JP);ХАРАДА Хиронори (JP);КУРОТАНИ Масахиро (JP);ТОДА Харухико (JP);САКАМОТО Кенитироу (JP) |
分类号 |
A61P9/00;A61P9/12;A61P43/00;C07D239/52 |
主分类号 |
A61P9/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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