发明名称 BICYCLIC PIPERAZINE COMPOUND AND USE THEREOF
摘要 <p>A compound represented by the formula (I) (wherein R&lt;1&gt; represents acyl; R&lt;2&gt; represents an optionally substituted hydrocarbon group, etc.; R&lt;3&gt; represents an optionally substituted hydrocarbon group, etc.; R&lt;4&gt; represents an optionally substituted hydrocarbon group, etc.; n is 0 to 4; and X represents oxygen, sulfur, etc.) or a salt of the compound. The compound has TGR23 antagonistic activity and is useful in the prevention of and treatments for cancers.</p>
申请公布号 WO2005021555(A1) 申请公布日期 2005.03.10
申请号 WO2004JP12683 申请日期 2004.08.26
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED;FUKATSU, KOHJI;NAKAYAMA, YUTAKA;TARUI, NAOKI;MORI, MASAAKI;MATSUMOTO, HIROKAZU;KURASAWA, OSAMU;BANNO, HIROSHI 发明人 FUKATSU, KOHJI;NAKAYAMA, YUTAKA;TARUI, NAOKI;MORI, MASAAKI;MATSUMOTO, HIROKAZU;KURASAWA, OSAMU;BANNO, HIROSHI
分类号 A61K31/55;A61K31/4985;A61K31/5377;A61K31/541;A61P1/14;A61P3/06;A61P3/10;A61P5/00;A61P5/14;A61P5/24;A61P9/12;A61P25/28;A61P35/00;A61P43/00;C07D487/04;C07D498/04;C07D513/04;(IPC1-7):C07D498/04;A61K31/537;A61K31/498 主分类号 A61K31/55
代理机构 代理人
主权项
地址